Fluorinated 1,3-benzothiazin-4-ones containing fluoroquinolone fragment

Chemistry of Heterocyclic Compounds - We have developed an efficient synthetic approach to potential antibacterial agents with double mechanism of action through the combination of antibacterial...     

Pericyclic reactions in the synthesis of new 5-aryl-5,6-dihydroquinolino[2,1-b]quinazolin-12-ones

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Synthesis of New Purine Derivatives Containing α- and ω-Amino Acid Fragments

Russian Journal of Organic Chemistry - New conjugates of purine and 2-aminopurine with several α- and ω-amino acids have been synthesized following two approaches based on the...     

Synthesis and antiherpetic activity of novel purine conjugates with 7,8-difluoro-3-methyl-3,4-dihydro-2H-1,4-benzoxazine

Chemistry of Heterocyclic Compounds - A method for the synthesis of novel purine conjugates with 7,8-difluoro-3-methyl-3,4-dihydro-2H-1,4-benzoxazine containing fragments of ω-amino acids with...     

Novel purine conjugates with N-heterocycles: synthesis and anti-influenza activity

Chemistry of Heterocyclic Compounds - A number of novel amides were synthesized by coupling of 6-[(9H-purin-6-yl)amino]hexanoic acid to heterocyclic amines. The antiviral activity of the obtained...     

Synthesis and antimycobacterial activity of purine conjugates with (S)-lysine and (S)-ornithine

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Three-component green synthesis of 6-ethoxycarbonyl-5-methyl-7-(thien-2-yl)-4,7-dihydro[1,2,4]triazolo[1,5-a]pyrimidine,a promising antituberculosis drug

Russian Chemical Bulletin - A new simple, technological, and environmentally friendly method for the catalyst-free synthesis in water of a promising antituberculosis drug,...     

Antiviral drug Triazavirin,selectively labeled with 2H, 13C,and 15N stable isotopes. Synthesis and properties

Chemistry of Heterocyclic Compounds - Isotope-labeled antiviral drug Triazavirin containing 2H, 13C, and 15N atoms in its structure has been synthesized. 13C2H3I and KS13CN served as donors of 13C...