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Late‐Stage Diversification of Peptides by Metal‐Free CH Arylation |
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| Authors: | Dipl‐Chem Yingjun Zhu Michaela Bauer Jasper Ploog Prof?Dr Lutz Ackermann |
| Institution: | Institut für Organische und Biomolekulare Chemie, Georg‐August‐Universit?t, Tammannstrasse 2, 37077 G?ttingen (Germany), Fax: (+49)?551‐39‐6777 |
| Abstract: | The bioorthogonal late‐stage diversification of functionalized oligopeptides was accomplished through a metal‐free, site‐selective C?H arylation of engineered indole derivatives under mild reaction conditions. |
| Keywords: | C H activation chemoselective reactions late stage diversification metal‐free reactions peptides |