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Intrinsic relative preference profile of pan-kinase inhibitor drug staurosporine towards the clinically occurring gatekeeper mutations in Protein Tyrosine Kinases
Affiliation:1. Department of Radiation Oncology, Stanford University, Palo Alto, California;2. Global Institution for Collaborative Research and Education, Hokkaido University, Sapporo, Japan;3. Stanford Cancer Institute, Stanford, California;1. Research and Development Division, OSAKA SODA Co., Ltd., Amagasaki, Hyogo 660-0842, Japan;2. Graduate School of Engineering, Osaka University, 2-1 Yamadaoka, Suita, Osaka 565-0871, Japan;1. Key Laboratory for Liquid–Solid Structural Evolution and Processing of Materials, Ministry of Education, Shandong University, Jinan 250061, China;2. School of Engineering, Edith Cowan University, 270 Joondalup Drive, Perth, WA 6027, Australia
Abstract:
Keywords:Protein tyrosine kinase  Pan-kinase inhibitor  Staurosporine  Gatekeeper mutation  Kinase context  Relative preference
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