Total Syntheses of the Chlorinated β‐Carboline Alkaloids Bauerine A,B, and C |
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| Authors: | Berthold Pohl Thomas Luchterhandt |
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| Institution: | Department of Pharmacy , Center for Drug Research, Ludwig‐Maximilians‐Universit?t , Munich, Germany |
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| Abstract: | The first total synthesis of the chlorinated 1‐oxo‐β‐carboline alkaloid bauerine C based on a Japp–Klingemann reaction is reported. An intermediate of this synthesis was converted to the fully aromatic β‐carboline bauerine B, and the related alkaloid bauerine A was prepared in an analogous manner. |
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| Keywords: | alkaloids bauerine cyclizations dehydrogenations 1‐oxo‐β‐carbolines |
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