Efficient Synthesis of Chiral 1,1′‐Sulfonyl Bisaziridines |
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| Authors: | Nawel Khettache Amel Bendjeddou Malika Berredjem Zine Regainia Veronique Montero Chantal Menut |
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| Institution: | 1. Laboratoire de Chimie Bioorganique , Université d'Annaba , Annaba, Algéria;2. Laboratoire de Chimie Biomoléculaire , Université Montpellier II , Montpellier Cedex, France |
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| Abstract: | An efficient three‐step synthesis of chiral 1,1′‐(sulfonyl)bisaziridines is described. Preparation of these compounds was carried out easily starting from N,N′‐sulfonyl bis‐(α‐L‐aminoester) to afford the title compounds in very good yields. These 1,1′‐(sulfonyl)bisaziridines can constitute interesting synthetic building blocks. |
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| Keywords: | Sulfonylbisaziridine sulfamide aziridine heterocycle |
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