| α-(1,3,4-噻二唑-5-基)氨基烃基膦酸酯的合成及生物活性 |
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| 引用本文： | 曹蕾,汪焱钢,宋新建,刘国华.α-(1,3,4-噻二唑-5-基)氨基烃基膦酸酯的合成及生物活性[J].有机化学,2005,25(8):1007-1010. |
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| 作者姓名： | 曹蕾 汪焱钢 宋新建 刘国华 |
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| 作者单位： | 1. 华中师范大学化学学院,武汉,430079;深圳市水质检测中心,深圳,518036
2. 华中师范大学化学学院,武汉,430079 |
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| 摘 要： | 以5-氨基-2-巯基的席夫碱与亚磷酸二乙酯反应, 合成了15个新的α-(1,3,4-噻二唑-5-基)氨基烃基膦酸酯, 初步的生物活性测试表明部分目标化合物具有较好的植物生长调节活性, 其中2,4-二氯苯甲醛、呋喃甲醛和吲哚甲醛的席夫碱生成的α-氨基烃基膦酸酯具有较好的生长素活性.
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| 关 键 词： | 噻二唑 席夫碱 膦酸酯 生物活性 植物生长调节剂 生长素 |
| 收稿时间： | 2004-10-25 |
| 修稿时间： | 2004年10月25 |
Synthesis and Biological Activity of α-(1,3,4-Thiadiazol-5-yl)-aminoalkyl Phosphonates |
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| CAO,Lei,WANG Yan-Gang,SONG Xin-Jian,LIU,Guo-Hua.Synthesis and Biological Activity of α-(1,3,4-Thiadiazol-5-yl)-aminoalkyl Phosphonates[J].Chinese Journal of Organic Chemistry,2005,25(8):1007-1010. |
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| Authors: | CAO Lei WANG Yan-Gang SONG Xin-Jian LIU Guo-Hua |
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| Institution: | ( College of Chemistry, Central China Normal University, Wuhan 430079)( Shenzhen Water Quality Centre, Shenzhen 518036) |
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| Abstract: | Fifteen new α-(1,3,4-thiadiazol-5-yl)aminoalkyl phosphonates have been synthesized by addition reaction of diethyl phosphite to the corresponding Schiff bases of 5-amino-2-mecapto-1,3,4-thiadiazole. Preliminarily biological activity tests show that some target compounds have good activity as plant growth regulator, particularly α-aminoalkyl phosphonates of 2,4-dichlorobenzaldehyde, furfuraldehyde and indolylaldehyde have better auxin activity. |
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| Keywords: | thiadiazole Schiff base phosphonate biological activity plant growth regulator auxin |
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