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Acidic pH‐Responsive siRNA Conjugate for Reversible Carrier Stability and Accelerated Endosomal Escape with Reduced IFNα‐Associated Immune Response
Authors:Hiroyasu Takemoto  Dr. Kanjiro Miyata  Shota Hattori  Dr. Takehiko Ishii  Tomoya Suma  Satoshi Uchida  Dr. Nobuhiro Nishiyama  Dr. Kazunori Kataoka
Affiliation:1. Department of Materials Engineering, The University of Tokyo, Hongo 7‐3‐1, Bunkyo‐ku, Tokyo 113‐8656 (Japan) http://www.bmw.t.u‐tokyo.ac.jp/;2. Division of Clinical Biotechnology, Center for Disease Biology and Integrative Medicine, The University of Tokyo, Hongo 7‐3‐1, Bunkyo‐ku, Tokyo 113‐0033 (Japan);3. Department of Bioengineering, The University of Tokyo, Hongo 7‐3‐1, Bunkyo‐ku, Tokyo 113‐8656 (Japan);4. Polymer Chemistry Division, Chemical Resources Laboratory, Tokyo Institute of Technology, R1‐11, 4259 Nagatsuta, Midori‐ku, Yokohama 226‐8503 (Japan)
Abstract:
Keywords:conjugation  drug delivery  drug design  polymers  siRNA
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