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Acylmethanesulfonamides as new acylating agents for primary amines |
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| Authors: | Silvia Coniglio Sandro Colagioia Fabrizio D'Alessandro Valerio D'Elia Valerie Orlando |
| Affiliation: | a Dompé Research and Development, Chemistry Department, Dompé S.p.A., Via Campo di Pile, 67100 L'Aquila, Italy b Dompé Research and Development, Analytical Department, Dompé S.p.A., Via Campo di Pile, 67100 L'Aquila, Italy |
| Abstract: | A new, simple and efficient procedure for the preparation of secondary amides through internal condensation of acylmethanesulfonamides ammonium salts is described. The selective acylation of mixed primary-secondary amines could be an attractive application of the new method. |
| Keywords: | Acylmethanesulfonamides Mixed primary-secondary amine Condensation reaction |
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