|
|||||
|
|
New synthesis of 3-substituted indoles using lithium trimethylsilyldiazomethane |
|
| Authors: | Takashi Miyagi |
| Institution: | Graduate School of Pharmaceutical Sciences, Nagoya City University, 3-1 Tanabe-dori, Mizuho-ku, Nagoya 467-8603, Japan |
| Abstract: | Lithium trimethylsilyldiazomethane smoothly reacted with N-tosyl-o-acylanilines to give 3-substituted indoles in good to high yields. |
| Keywords: | o-Acylanilines Alkylidene carbene Indoles Intramolecular N-H insertion Trimethylsilyldiazomethane |
| 本文献已被 ScienceDirect 等数据库收录！ | |