| O-烷基O-取代苯基硫代磷酰胺酯类化合物的合成及其结构与杀虫活性的定量关系 |
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| 引用本文： | 陈茹玉,王惠林,曹如珍,张政朴,邵久书,朱兰惠,陈学仁,杨华铮. O-烷基O-取代苯基硫代磷酰胺酯类化合物的合成及其结构与杀虫活性的定量关系[J]. 高等学校化学学报, 1987, 8(8): 706 |
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| 作者姓名： | 陈茹玉 王惠林 曹如珍 张政朴 邵久书 朱兰惠 陈学仁 杨华铮 |
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| 作者单位： | 南开大学元素有机化学研究所 |
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| 摘 要： | 合成了19种O-烷基O-取代苯基硫代磷酰胺酯类化合物,在定量测定其杀虫活性的基础上,对该类化合物进行了结构与活性定量关系的解析。结果表明,分子中芳基上取代基的电子效应与2,3-位上取代基的疏水性质对活性有重要影响。
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| 收稿时间： | 1986-03-26 |
Quantitative Structure-Activity Study on a Series of Insecticidal O-Alkyl O-Aryl Phosphoramidothioates |
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| Chen Ruyu,Wang Huilin,Cao Ruzhen,Zhang Zhengpu,Shao Jiushu,Zhu Lanhui,Chen Xueren,Yang Huazheng. Quantitative Structure-Activity Study on a Series of Insecticidal O-Alkyl O-Aryl Phosphoramidothioates[J]. Chemical Research In Chinese Universities, 1987, 8(8): 706 |
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| Authors: | Chen Ruyu Wang Huilin Cao Ruzhen Zhang Zhengpu Shao Jiushu Zhu Lanhui Chen Xueren Yang Huazheng |
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| Affiliation: | Institute of Elemento-Organic Chemistry, Nan(?) University, Tianjin |
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| Abstract: | 19 O-Alkyl O-aryl phosphoramidothioates were synthesized by the reaction of O-alkyl O-aryl phosphorochloridothioates with aqueous ammonia and the quantitative relationship between their structures and insecticidal activities was analyzed using physicochemical parameters of the substituents in the benzene ring by regression analysis. It was found that the electronic and hydrophobic effects of the substituents are important to the activity. |
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