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Targeting Matrix Metalloproteinases: Design of a Bifunctional Inhibitor for Presentation by Tumour‐Associated Galectins
Authors:Dr Marco Bartoloni  Dr Blanca E Domínguez  Dr Elisa Dragoni  Dr Barbara Richichi  Dr Marco Fragai  Dr Sabine André  Prof Hans‐Joachim Gabius  Dr Ana Ardá  Prof Claudio Luchinat  Prof Jesús Jiménez‐Barbero  Prof Cristina Nativi
Institution:1. Department of Chemistry, University of Florence, Via della Lastruccia, 13 50019 Sesto F.no Firenze (Italy);2. Centro de Investigationes Biològicas, CSIC, Ramiro de Maetzu 9, 28040 Madrid (Spain);3. Centro de Investigaciones Químicas, Universidad Autónoma del Estado de Morelos, Av. Universidad 1001, 62210, Cuernavaca, Morelos (México);4. CERM, University of Florence, Via Sacconi, 6 50019 Sesto F.no Firenze (Italy);5. Institute of Physiological Chemistry, Faculty of Veterinary Medicine, Ludwig‐Maximilians‐University, Veterin?rstr. 13, 80539 München (Germany)
Abstract:
Keywords:glycoconjugates  inhibitors  ligand design  metalloproteins  NMR spectroscopy
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