Direct C-arylation of beta-enamino esters and ketones with arynes |
| |
| Authors: | Ramtohul Yeeman K Chartrand Anik |
| |
| Institution: | Department of Medicinal Chemistry, Merck Frosst Centre for Therapeutic Research, Merck Frosst Canada & Co. Inc., P.O. Box 1005, 16711 Trans Canada Highway, Kirkland, Quebec, Canada H9H 3L1. yeeman_ramtohul@merck.com |
| |
| Abstract: | An efficient, mild, and general method for the C-arylation of beta-enamino esters and ketones with arynes has been developed. This methodology provides a facile and direct access to a variety of substituted aromatic beta-enamino compounds in moderate to excellent yield. reaction: see text] |
| |
| Keywords: | |
| 本文献已被 PubMed 等数据库收录！ |
|
