| Direct C–H amination for indole synthesis from N-Ts-2-Styrylaniline derivatives catalyzed by copper salt |
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| 作者姓名： | Di Chen Han-Jie Mo Ding-Ben Chen Jian-Guo Yang |
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| 作者单位： | School of Pharmaceutical and Chemical Engineering, Taizhou University, Taizhou 317000, China |
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| 基金项目： | This work was financially supported by the National Natural Science Foundation of China (Nos. 21272169, 21302135), the Key Innovation Team of Science & Technology in Zhejiang Province (No. 2010R50018-10), the Science and Technology Bureau of Taizhou (No. 08KY10) and the Key Disciplines of Applied Chemistry of Zhejiang Province, Taizhou University. |
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| 摘 要： | A direct C–H amination reaction of N-Ts-2-Styrylaniline derivatives to realize the synthesis of indole derivatives was developed in the presence of copper salt. A variety of N-Ts-2-Styrylaniline derivatives were transformed into the corresponding indole products in good to excellent yield under mild conditions with the oxidation of potassium persulfate.
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Direct C-H amination for indole synthesis from N-Ts-2-Styrylaniline derivatives catalyzed by copper salt |
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| Di Chen,Han-Jie Mo,Ding-Ben Chen,Jian-Guo Yang.Direct C-H amination for indole synthesis from N-Ts-2-Styrylaniline derivatives catalyzed by copper salt[J].Chinese Chemical Letters,2015,26(8):969-972. |
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| Authors: | Di Chen Han-Jie Mo Ding-Ben Chen Jian-Guo Yang |
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| Institution: | School of Pharmaceutical and Chemical Engineering, Taizhou University, Taizhou 317000, China |
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| Abstract: | A direct C-H amination reaction of N-Ts-2-Styrylaniline derivatives to realize the synthesis of indole derivatives was developed in the presence of copper salt. A variety of N-Ts-2-Styrylaniline derivatives were transformed into the corresponding indole products in good to excellent yield under mild conditions with the oxidation of potassium persulfate. |
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| Keywords: | C-H amination N-Ts-2-Styrylaniline derivatives Indole Copper salt Potassium persulfate |
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