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Preparation of 7-aminoquinolines as candidate antiparasitic agents
Authors:Anica Markovac  Geng-Shuen Wu  Maurice P. Lamontagne  Peter Blumbergs  Ao Meng-Sheng
Abstract:A series of ten 7-quinolinediamines were prepared and evaluated for potential antiparasitic activity against P. berghei, P. cynomolgi, L. donovani and T. rhodesiense. Compounds 1d and 8 showed activity being slightly effective against L. donovani in hamsters.
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