A simple and efficient route to β-substituted pyrroles |
| |
| Authors: | Joshua Rokach Pierre Hamel Masatoshi Kakushima Graham M. Smith |
| |
| Affiliation: | Merck Frosst Laboratories, P.O. Box 1005, Pointe-Claire/Dorval, Québec, Canada H9R 4P8;Merck Sharp & Dohme Research Laboratories, P.O. Box 2000, Rahway, NJ 07065 U.S.A. |
| |
| Abstract: | -Phenylsulfonylpyrrole undergoes Friedel-Crafts acylation exclusively at the β-position of the pyrrole ring, thus allowing a simple and efficient synthesis of β-acylated pyrroles. |
| |
| Keywords: | |
| 本文献已被 ScienceDirect 等数据库收录！ |
|
