Transition metal catalyzed synthesis of 5-azaindoles |
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| Affiliation: | 1. Department of Drug Sciences and Health Products, University of Messina, Viale Annunziata, 98168 Messina, Italy;2. Institute of Pharmacy and Biochemistry, University of Mainz, Staudinger Weg 5, D-55099 Mainz, Germany;3. Department of Pharmaceutical Sciences, University of Milan, Via Mangiagalli 25, 20122 Milan, Italy;4. Department of Chemistry and Pharmacy, University of Sassari, Via Vienna 2, 07100 Sassari, Italy;5. Department of Chemical and Geological Sciences, University of Cagliari, S.S. 554, 09042 Monserrato, CA, Italy;6. Department of Chemistry and Industrial Chemistry, via Risorgimento 35, 56126 Pisa, Italy;7. Laboratory of “Metals in Medicine” (METMED), Department of Chemistry “Ugo Schiff”, University of Florence, Via della Lastruccia 3, Sesto Fiorentino, 50019 Firenze, Italy |
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| Abstract: | In an effort to develop synthetic procedures for the preparation of 2-substituted 5-azaindoles, the synthesis and cyclization reactions of acetylenic aminopyridines was explored. A novel method for the synthesis of 2-substituted 5-azaindoles via a transition metal catalyzed reaction is described. |
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