Recherches sur la formation et la transformation des esters LXXV[1]. Amines,amino-alcools et aminoalcoyl-monoesters des acides orthophosphorique et sulfurique: thiocarbamylation par l'isothiocyanate d'o-méthoxycarbonylphényle sans ou avec cyclisation intramoléculaire |
| |
Authors: | Emile Cherbuliez B. Willhalm O. Espejo S. Jaccard J. Rabinowitz |
| |
Abstract: | o-Methoxycarbonyl-phenylisothiocyanate V and primary alkylamines (R″? NH2) reacted in the appropriate medium yield the corresponding 2-mercapto-3-alkyl-3, 4-dihydro-quinazolinone-4 derivatives VI (the ? NH2 group is thiocarbamoylated by the ? N?C?S group and then acylated in an intramolecular reaction by the ? COOCH3 group with elimination of CH3OH). |
| |
Keywords: | |
|