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Phenylboronic acid as a mild and efficient catalyst for Biginelli reaction |
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| Authors: | Abdelmadjid Debache Ali Belfaitah Bertrand Carboni |
| Institution: | a Laboratoire des produits naturels d’origine végétale et de synthèse organique, Département de Chimie, Faculté des Sciences, Université Mentouri de Constantine, 25000 Constantine, Algeria b Sciences Chimiques de Rennes, UMR 6226 CNRS-Université de Rennes 1, Campus de Beaulieu, 35042 Rennes Cedex, France |
| Abstract: | The synthesis of 3,4-dihydropyrimidinone derivatives was achieved in good to excellent yields using phenylboronic acid as catalyst to promote the Biginelli three-component condensation of a diversity of aromatic aldehydes, ethyl acetoacetate and urea or thiourea. |
| Keywords: | Biginelli Boronic acid 3 4-Dihydropyrimidinone Three-component condensation |
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