An efficient electrophilic N-amination utilizing in situ generated chloramine under phase transfer conditions |
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| Authors: | Apurba Bhattacharya Nitin C Patel Michael Peddicord Luca Parlanti John A Grosso |
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| Institution: | a Department of Chemistry, Texas A&M University-Kingsville, Kingsville, TX 78363, United States
b Bristol-Myers Squibb Company, Process Research and Development Department, PO Box 191, New Brunswick, NJ 08903-0191, United States |
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| Abstract: | An efficient, one-pot, phase transfer N-amination technology was developed. The protocol utilizes chloramine, an inexpensive and safe electrophilic aminating agent potentially viable for commercial manufacturing. |
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