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In vitro antimicrobial evaluation and in silico studies of coumarin derivatives tagged with pyrano-pyridine and pyrano-pyrimidine moieties as DNA gyrase inhibitors
Authors:Fayed  Eman A  Nosseir  Eman S  Atef  Ahmed  El‑Kalyoubi  Samar A
Institution:1.Pharmaceutical Organic Chemistry Department, Faculty of Pharmacy (Girls), Al-Azhar University, Nasr City, 11754, Cairo, Egypt
;2.Pharmaceutical Medicinal Chemistry Department, Faculty of Pharmacy (Girls), Al-Azhar University, Nasr City, 11754, Cairo, Egypt
;3.Department of Microbiology, Regional Center of Mycology and Biotechnology, Al-Azhar University, Nasr City, Cairo, Egypt
;
Abstract:Molecular Diversity - Several coumarin-containing substitute nitrogen heterocycles have recently received considerable importance due to their diverse pharmacological properties. One-pot and rapid...
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