Diastereoselective reaction of (1S,2S)-2-amino-1-(4-nitrophenyl)-1,3-propanediol with aromatic aldehydes. Synthesis of (1R,2R,4S,5S,8S)-2,8-diaryl-4-(4-nitrophenyl)-1-aza-3,7-dioxabicyclo[3.3.0]octanes |
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| Authors: | M Madesclaire P Coudert V Gaumet V P Zaitsev Yu V Zaitseva |
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| Institution: | (1) School of Pharmacy, University of Auvergne, 28 Place Henri Dunant, Clermont-Ferrand, France;(2) Samara State University, Samara, 443011, Russia |
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| Abstract: | We have synthesized a series of (1R,2R,4S,5S,8S)-2,8-diaryl-4-(4-nitrophenyl)-1-aza-3,7-dioxabicyclo3.3.0]octanes as a result
of reaction of (1S,2S)-2-amino-1-(4-nitrophenyl)-1,3-propanediol with aromatic aldehydes. The structure of the compounds obtained
was established on the basis of 1H NMR data.
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Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 5, pp. 757–763, May, 2006. |
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| Keywords: | (1S 2S)-2-amino-1-(4-nitrophenyl)-1 3-propanediol (1R 2R 4S 5S 8S)-2 8-diaryl-4-(4-nitrophenyl)-1-aza-3 7-dioxabicyclo[3 3 0]octane oxazolidine diastereoselectivity 1H NMR |
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