|
|||||
|
|
Variations of the P2 group in HIV-1 protease inhibitors containing a tertiary alcohol in the transition-state mimicking scaffold |
|
| Authors: | Ekegren Jenny K Gising Johan Wallberg Hans Larhed Mats Samuelsson Bertil Hallberg Anders |
| Affiliation: | Department of Medicinal Chemistry, Organic Pharmaceutical Chemistry, BMC, Uppsala University, Box 574, SE-751 23, Uppsala, Sweden. |
| Abstract: | A short synthetic protocol leading to HIV-1 protease inhibitors with a tertiary alcohol based transition-state mimicking unit and different P2 side chains has been developed. |
| Keywords: | |
| 本文献已被 PubMed 等数据库收录！ | |