Abstract: | A new class of benzazolyl azolyl sulfamoyl acetamides was prepared from azolyl sulfamoyl acetates and benzazolyl amines in the presence of KOtBu in tetrahydrofuran. Compounds with benzothiazole‐thiazole, benzimidazole‐thiazole, benzothiazole‐imidazole, and benzimidazole‐imidazole moieties exhibited excellent antibacterial activity against Bacillus subtilis. |