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Palladium‐catalyzed regioselective C2‐arylation of 5‐aminoindole |
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| Authors: | Yunus Taskesenligil Ferruh Lafzi Haydar Kilic Nurullah Saracoglu |
| Abstract: | Pd(II)‐catalyzed C‐H arylations of 5‐aminoindole using iodobenzenes as aryl source was studied. Despite pivalamide directing group at 5‐position of the indole, the direct C2‐arylation of the indole observed in high yields and with high regioselectivity. |
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