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Vascular endothelial growth factor receptor-2 (VEGFR-2) inhibitors: development and validation of predictive 3-D QSAR models through extensive ligand- and structure-based approaches
Authors:Rino Ragno  Flavio Ballante  Adele Pirolli  Richard B Wickersham III  Alexandros Patsilinakos  Stéphanie Hesse  Enrico Perspicace  Gilbert Kirsch
Institution:1. Rome Center for Molecular Design, Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza Università di Roma, P. le A. Moro 5, 00185, Rome, Italy
2. Magma Dynamics srl, Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza Università di Roma, P. le A. Moro 5, 00185, Rome, Italy
3. Department of Biochemistry and Molecular Biophysics, Washington University in St. Louis School of Medicine, 700 South Euclid Avenue, St. Louis, MO, 63110, USA
4. SRSMC UMR CNRS7565 (former LIMBP), 1 Boulevard Arago, 57070, Metz, France
5. Genfit, Parc Eurasanté, 885 Avenue Eugène Avinée, 59120, Loss, France
Abstract:
Keywords:
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