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Synthesis of 4-azacyclopent-2-enones and 5,5-dialkyl-4-azacyclopent-2-enones
Authors:Jérôme Dauvergne  Vasudev Jadhav  Marie-Christine Matos  Michael R Pitts  Sanjay K Singh  John Whittall
Institution:a Charterhouse Therapeutics Ltd, Robert Robinson Building, University of Liverpool, Liverpool L69 7ZD, UK
b Stylacats Ltd, Development Labs, Cheshire Manufacturing Park, Ellesmere Port, Cheshire, UK
c Stylacats Ltd, Research Labs, Robert Robinson Building, University of Liverpool, Liverpool L69 7ZD, UK
Abstract:Three different methods are reported for the preparation of 4-azacyclo-2-enones 1, two of which allow the preparation of the compounds in optically active form. In addition, a facile route to 4-aza-5,5-dimethylcyclopent-2-enones 2 is disclosed.
Keywords:4-Aza-cyclopentenones  4-Aza-cyclopent-2-en-1-ols  Asymmetric synthesis of aminocyclopentenols  Lipase resolution
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