A Simple,Efficient Synthesis of N6-[bis(ethylamino) methylene]-N2-[(1,1-dimethylethoxy)carbonyl]-lysine (Boc-diethylhomoarginine) |
| |
| Authors: | H. B. Arzeno W. Bingenheimer D. J. Morgans Jr. |
| |
| Affiliation: | Institute of Organic Chemistry Syntex Research , 3401 Hillview Avenue, Palo Alto, CA, 94303 |
| |
| Abstract: | The synthesis of N6-(bis(ethylamino)methylene]-N2-[(1,1-dimethyl ethoxycarbonyl] lysine (Boc-diethylhomoarginine) by regiospecific amidination of lysine with (ethylamino) (ethylimino)-methanesulfonic acid (2) is described. |
| |
| Keywords: | |
|
|
