A Short Synthesis of 4- and 6-Azaindol-2(3H)-ones |
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Authors: | R. W. Daisley J. R. Hanbali |
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Affiliation: | Department of Pharmacy , Brighton Polytechnic , Moulsecoomb, Brighton, Sussex, BN2 4GJ, England |
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Abstract: | Although indol-2(3H)-ones possess a wide range of pharmacological1 and microbiological2 activities, the corresponding azaindol-2(3H)-ones have stimulated little interest. Successful syntheses have been reported for the title compounds3,4 involving several stages which in our hands gave a variety of side products, especially in the hydrogenation stage. |
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