Original synthesis of 2-substituted-4,11-dimethoxy-1-(phenylsulfonyl)-2,3-dihydro-1H-naphtho[2,3-f]indole-5,10-diones using TDAE and Cu-catalyzed reaction strategy |
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| Authors: | Omar KhoumeriGamal Giuglio-Tonolo Maxime D CrozetThierry Terme Patrice Vanelle |
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| Institution: | Laboratoire Chimie Provence LCP, UMR CNRS 6264, Universités d’Aix-Marseille I, II et III, Equipe Pharmaco-Chimie Radicalaire, Faculté de Pharmacie, 27 Boulevard Jean Moulin, 13385 Marseille Cedex 05, France |
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| Abstract: | We report herein an original and rapid synthesis of 2-substituted-4,11-dimethoxy-1-(phenylsulfonyl)-2,3-dihydro-1H-naphtho2,3-f]indole-5,10-diones by TDAE mediated synthesis of N-benzylsulfonamides followed by an intramolecular N-arylation using Cu-catalyzed system. |
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| Keywords: | TDAE N-(Benzenesulfonyl)benzylimine Cu-catalyzed reaction Naphtho[2 3-f]indole-5 10-dione |
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