A facile transformation of bicyclic keto esters to bisprotected (±)-8-epithienamycin <span class="math"><math><mtext>via</mtext></math></span> enol activation期刊界 All Journals 搜尽天下杂志传播学术成果专业期刊搜索期刊信息化学术搜索

A facile transformation of bicyclic keto esters to bisprotected (±)-8-epithienamycin $via$ enol activation

Authors:	M. Sletzinger T. Liu R.A. Reamer I. Shinkai

Affiliation:	Merck Sharp & Dohme Research Laboratories, Division of Merck & Co., Inc., Rahway, New Jersey, 07065, U.S.A.

Abstract:	A facile “one-pot” transformation of bicyclic keto ester (2) to bisprotected (±)-8-epithienamycin $via$ enol phosphate activation followed by the addition-elimination reaction of $N$ -protected cysteamine derivative is described.

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