A one-pot asymmetric organocatalytic tandem reaction for the synthesis of oxazine derivatives |
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| Authors: | Jin Zhichao Yu Feng Wang Xiao Huang Huicai Luo Xiaoyan Liang Xinmiao Ye Jinxing |
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| Affiliation: | Engineering Research Centre of Pharmaceutical Process Chemistry, Ministry of Education, School of Pharmacy, East China University of Science and Technology, 130 Meilong Road, Shanghai 200237, China. |
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| Abstract: | An easy one-pot tandem reaction catalyzed by a chiral secondary amine for the synthesis of optically active oxazine derivatives has been performed and the corresponding substituted benzo[d]pyrido[2,1-b][1,3]oxazine derivatives were afforded in generally high yields (up to 99%) and excellent enantioselectivities (up to >99%). |
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