Chan-Lam-type S-arylation of thiols with boronic acids at room temperature |
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Authors: | Xu Hua-Jian Zhao Yong-Qiang Feng Teng Feng Yi-Si |
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Affiliation: | School of Medical Engineering, Hefei University of Technology, Hefei 230009, P. R. China. hjxu@hfut.edu.cn |
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Abstract: | In this work, an efficient CuSO(4)-catalyzed S-arylation of thiols with aryl and heteroaryl boronic acids at room temperature is established. This catalytic system can tolerate a wide variety of thiols and arylboronic acids in the presence of only 5 mol % of CuSO(4) as the catalyst and inexpensive 1,10-phen·H(2)O as the ligand. Moreover, this catalytic system used environment-friendly solvent (EtOH) and oxidant (oxygen). |
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