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Substrate-Selective Inhibition of Protein Kinase PDK1 by Small Compounds that Bind to the PIF-Pocket Allosteric Docking Site
Authors:Katrien Busschots  Laura A Lopez-Garcia  Carmen Lammi  Adriana Stroba  Stefan Zeuzem  Albrecht Piiper  Pedro M Alzari  Sonja Neimanis  Jose M Arencibia  Matthias Engel  Jörg O Schulze  Ricardo M Biondi
Institution:1. Research Group PhosphoSites, Department of Internal Medicine I, Universitätsklinikum Frankfurt, Theodor-Stern-Kai 7, 60590 Frankfurt, Germany;2. Research Group PhosphoSites, Department of Pharmaceutical and Medicinal Chemistry, University of Saarland, 66041 Saarbrücken, Germany;3. Structural Biochemistry Unit, Pasteur Institute, Rue du Dr. Roux 25, F-75724 Paris, France
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