Abstract: | Amidoalkylation of three benzoheterocycles, benzimidazole-2-one, 1,3-dihydrobenzoc]-thiophene 2,2-dioxide and 1,3-dihydro-2,1,3-benzothiadiazole using N-acylhippuric acids was successful. The corresponding phenylglycine analogs were prepared by removal of the N-acyl protecting group. |