Synthesis of substituted 2-cyanoarylboronic esters |
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| Authors: | Lysén Morten Hansen Henriette M Begtrup Mikael Kristensen Jesper L |
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| Affiliation: | Department of Medicinal Chemistry, Danish University of Pharmaceutical Sciences, Universitetsparken 2, DK-2100 Copenhagen, Denmark. |
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| Abstract: | The synthesis of substituted 2-cyanoarylboronic esters is described via lithiation/in situ trapping of the corresponding methoxy-, trifluoromethyl-, fluoro-, chloro-, and bromobenzonitriles. The crude arylboronic esters were obtained in high yields and purities and with good regioselectivities. |
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