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Polymer‐Supported Hypervalent Iodine Reagent Mediated Synthesis of α‐Azidoketones |
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| Authors: | Huey‐Min Wang Rei‐Sheu Hou Jian‐Long Wu Ling‐Ching Chen |
| Affiliation: | 1. Chung Hwa University of Medical Technology, Tainan 717, Taiwan, R.O.C.;2. Graduate Institute of Pharmaceutical Sciences, College of Pharmacy, Kaohsiung Medical University, Kaohsiung 807, Taiwan, R.O.C. |
| Abstract: | The reaction of aryl ketones with sodium azide using polymer‐supported bis(trifluoroacetoxyiodo)‐benzene (PSBTI) in the presence of trifluoroacetic acid (TFA) to prepare α‐azidoketones in one‐pot conditions is reported. |
| Keywords: | Hypervalent iodine Polymer‐supported bis(trifluoroacetoxyiodo)benzene α ‐Azidoketones |