Selective mono-arylation in palladium-catalyzed cross-coupling reaction of dichlorotriazines with phenylboronate ester derivatives |
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| Authors: | Jin-Fu Dong Xin Yu Cheng-Qing Ning Liang Hu Nie-Fang Yu |
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| Affiliation: | 1. School of Pharmaceutical Sciences, Central South University, Changsha 410013, China
2. School of Pharmaceutical Sciences,Sun Yat-sen University, Guangzhou 51006, China |
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| Abstract: | Palladium-catalyzed cross-coupling reaction between dichlorotriazines and phenylboronate esters produced the mono-arylated triazines selectively and thus, the corresponding phenyltriazine derivatives could be assembled efficiently in moderate to good overall yields (50–80%). |
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| Keywords: | Suzuki cross-coupling reaction Dichlorotriazines Aryl boronic esters Pd(PPh3) |
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