Synthetic route to chiral tetrahydroquinoxalines via ring-opening of activated aziridines |
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| Authors: | Ghorai Manas K Sahoo Ashis K Kumar Sarvesh |
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| Affiliation: | Department of Chemistry, Indian Institute of Technology, Kanpur 208016, India. |
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| Abstract: | A highly regio- and stereoselective route for the synthesis of racemic and nonracemic tetrahydroquinoxalines via the S(N)2-type ring-opening of activated aziridines with 2-bromoanilines followed by the Pd-catalyzed intramolecular C-N bond formation is described. |
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