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Heteroaromatic Tosylates as Electrophiles in Regioselective Mizoroki–Heck‐Coupling Reactions with Electron‐Rich Olefins |
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| Authors: | Thomas M Gøgsig Anders T Lindhardt Dr Mouloud Dekhane Dr Julie Grouleff Troels Skrydstrup Prof Dr |
| Institution: | 1. The Center for Insoluble Protein Structures (inSPIN), Department of Chemistry and the Interdisciplinary Nanoscience Center, Aarhus University, Langelandsgade 140, 8000 Aarhus (Denmark), Fax: (+45)?8619‐6199;2. AstraZeneca, Business park, Charter Way, Macclesfield, Cheshire, SK10 2NA (UK) |
| Abstract: | Easy and direct : Regioselective Mizoroki–Heck‐coupling reactions using heteroaromatic tosylates as electrophiles were achieved, thus providing direct and easy access to highly functionalized α‐heteroarylvinyl amides and ethers.  |
| Keywords: | aryl tosylates C?C coupling Mizoroki– Heck coupling heterocycles palladium |