| Tandem Approach to Functionalized Pyrrolo[3,4-α]carbazole-1,3-diones via a Pd-catalyzed Indole-to-carbazole Transformation |
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| 作者姓名： | GUO Lianghua XU Mei JIAN Yong LIU Sheng PAN Weidong DUAN Lian |
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| 作者单位： | State Key Laboratory of Functions and Applications of Medicinal Plants |
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| 基金项目： | the National Natural Science Foundation of China;the Science Foundation of Guizhou Province,China |
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| 摘 要： | A one-pot and efficient tliree-component reaction of indoles, acrylates and maleimides for the synthesis of pyrrolo3,4-α]carbazole-1,3-dione derivatives was developed. Three C-C bonds and one ring were created in a single step via an indole-to-carbazole transformation triggered by Pd(II)-catalyzed direct C3-alkenylation of indoles.
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| 关 键 词： | CARBAZOLE One-pot TANDEM REACTION Three-component REACTION Indole-to-carbazole |
| 收稿时间： | 2018-12-21 |
Tandem Approach to Functionalized Pyrrolo[3,4-a]carbazole-1,3-diones via a Pd-catalyzed Indole-to-carbazole Transformation |
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| GUO Lianghua,XU Mei,JIAN Yong,LIU Sheng,PAN Weidong,DUAN Lian.Tandem Approach to Functionalized Pyrrolo[3,4-a]carbazole-1,3-diones via a Pd-catalyzed Indole-to-carbazole Transformation[J].Chemical Research in Chinese University,2019,35(4):621-626. |
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| Authors: | GUO Lianghua XU Mei JIAN Yong LIU Sheng PAN Weidong DUAN Lian |
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| Institution: | State Key Laboratory of Functions and Applications of Medicinal Plants, Guizhou Medical University, Guiyang 550014, P. R. China |
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| Abstract: | A one-pot and efficient three-component reaction of indoles, acrylates and maleimides for the synthesis of pyrrolo3,4-a]carbazole-1,3-dione derivatives was developed. Three C-C bonds and one ring were created in a single step via an indole-to-carbazole transformation triggered by Pd(Ⅱ)-catalyzed direct C3-alkenylation of indoles. |
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| Keywords: | Carbazole One-pot Tandem reaction Three-component reaction Indole-to-carbazole |
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