1. Faculty of Chemistry, University of Warsaw, Pasteura 1, 02-093 Warszawa, Poland;2. National Drug Institute, Che?mska 30/34, 00-725 Warszawa, Poland
Abstract:
A mild and efficient method for the synthesis of fulgimides is presented in which the peptide coupling reagent BOP is employed for dehydratation of fulgenic acid monoamides (succinamic acids). The disclosed method proved to be superior to those described in the literature.