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Palladium‐Catalyzed Construction of Amidines from Arylboronic Acids under Oxidative Conditions |
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| Authors: | Fengxiang Zhu Yahui Li Zechao Wang Prof Dr Romano V A Orru Prof Dr Bert U W Maes Prof Dr Xiao‐Feng Wu |
| Institution: | 1. Leibniz-Institut für Katalyse e.V. an der, Universit?t Rostock, Rostock, Germany;2. Department of Chemistry and Pharmaceutical Sciences and Amsterdam, Institute for Molecules, Medicines and Systems (AIMMS), VU University, Amsterdam, Amsterdam, The Netherlands;3. Department of Chemistry, University of Antwerp, Antwerp, Belgium |
| Abstract: | A valuable palladium‐catalyzed three‐component coupling reaction for the synthesis of amidines has been developed. Using arylboronic acids, isocyanides, and anilines as the reactants under oxidative conditions, various amidines were isolated in good yields with good functional group tolerances. |
| Keywords: | amidines boronic acids domino reaction isocyanides palladium |