|
|||||
|
|
A facile and environmental friendly strategy for the synthesis of N-methoxyquinolin-2(1H)-ones |
|
| Authors: | Xianying Gao Apeng Liang Jingya Li Dapeng Zou Yangjie Wu Yusheng Wu |
| Institution: | 1. The College of Chemistry and Molecular Engineering, Zhengzhou University, Zhengzhou 450052, PR China;2. Collaborative Innovation Center of New Drug Research and Safety Evaluation, Henan Province, PR China;3. Tetranov Biopharm, LLC., No.75 Daxue Road, Zhengzhou 450052, PR China;4. Tetranov International, Inc., 100 Jersey Avenue, Suite A340, New Brunswick, NJ 08901, USA |
| Abstract: | A facile and environmental friendly protocol for the construction of N-methoxyquinolin-2(1H)-ones was developed using a stable and easily available N-methoxyquinoline-1-ium tetrafluoroborate as starting material. Due to the mild reaction conditions, a broad range of N-methoxyquinolin-2(1H)-ones with different functional groups have been prepared in reasonable yields. |
| Keywords: | N-methoxyquinolin-2(1H)-ones N-methoxyquinoline-1-ium tetrafluoroborate salts N-protected |
| 本文献已被 ScienceDirect 等数据库收录！ | |