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Palladium-catalyzed direct ortho-acylation through an oxidative coupling of 2-arylbenzothiazoles with benzylic alcohols |
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| Authors: | Qiuping Ding Huafang Ji Changqing YeJiajia Wang Junyan WangLiyun Zhou Yiyuan Peng |
| Institution: | Key Laboratory of Functional Small Organic Molecules, Ministry of Education and College of Chemistry & Chemical Engineering, Jiangxi Normal University, Nanchang, Jiangxi 330022, China |
| Abstract: | An efficient protocol was developed for Pd-catalyzed direct C–H bond acylation by cross-dehydrogenative-coupling of arylbenzothiazoles and benzylic alcohols using tert-butyl hydroperoxide (TBHP) as the oxidant. The acylation reactions exhibit good reactivities and excellent regioselectivity. |
| Keywords: | ortho-Acylation 2-Arylbenzothiazoles Benzylic alcohols tert-Butyl hydroperoxide |
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