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A mild and efficient new synthesis of aryl sulfones from boronic acids and sulfinic acid salts |
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| Authors: | Christian Beaulieu Daniel Guay David A. Evans |
| Affiliation: | a Department of Medicinal Chemistry, Merck Frosst Centre for Therapeutic Research, PO Box 1005, Pointe-Claire-Dorval, Québec, Canada H9R 4P8 b Department of Chemistry and Chemical Biology, Harvard University, 12 Oxford Street, Cambridge MA 02138, USA |
| Abstract: | A new efficient and mild preparation of sulfones from boronic acids and sulfinic acid salts is reported. The cross-coupling reaction mediated by cupric acetate gives access to a variety of sulfones in excellent yield. |
| Keywords: | Aryl sulfone Cross-coupling reaction Boronic acid |
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