Ruthenium‐Catalyzed C7 Amidation of Indoline CH Bonds with Sulfonyl Azides |
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| Authors: | Changduo Pan Ablimit Abdukader Jie Han Prof. Dr. Yixiang Cheng Prof. Dr. Chengjian Zhu |
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| Affiliation: | 1. State Key Laboratory of Coordination Chemistry, School of Chemistry and Chemical Engineering, Nanjing University, Nanjing, 210093 (P.R. China);2. Wenzhou Institute of Industry & Science, Wenzhou 325000 (P.R. China) |
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| Abstract: | A ruthenium‐catalyzed direct C7 amidation of indoline C?H bonds with sulfonyl azides was developed. This procedure allows the synthesis of a variety of 7‐amino‐substituted indolines, which are useful in pharmaceutical. The good functional tolerances, as well as the mild conditions, are prominent feature of this method. |
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| Keywords: | amidation C H activation indolines ruthenium sulfonyl azides |
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