Novel synthesis of C-3-(hetero)aryl [1,2,3]triazolo[1,5-a]pyridines using the Stille reaction |
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| Authors: | Hervé GermainCraig S. Harris,Honorine Lebraud |
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| Affiliation: | AstraZeneca, Centre de Recherches, Z.I. la Pompelle, BP1050, 51689 Reims Cedex 2, France |
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| Abstract: | Herein, we report a novel and high yielding approach for the preparation of the first C-3-organometallic substituted [1,2,3]triazolo[1,5-a]pyridine and its application to the Stille reaction using MAOS. |
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| Keywords: | [1,2,3]Triazolo[1,5-a]pyridine Stille cross-coupling reaction Microwave-assisted organic synthesis (MAOS) |
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