Reactivity study of 1H-thieno[3,2-d][1,3]oxazine-2,4-dione toward the synthesis of bicyclic 3,4-dihydro-1H-thieno[3,2-e][1,4]diazepine-2,5-dione analogues |
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| Authors: | Brouillette Yann Lisowski Vincent Fulcrand Pierre Martinez Jean |
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| Affiliation: | Laboratoire des Aminoacides, Peptides et Protéines (LAPP), CNRS UMR 5810, UMI-UMII, UFR des Sciences Pharmaceutiques et Biologiques, 15 Avenue Charles Flahault, 34093 Montpellier Cedex 5, France. |
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| Abstract: | A series of 10 optically pure 3,4-dihydro-1H-thieno[3,2-e][1,4]diazepine-2,5-dione derivatives has been synthesized in 41-75% yields on treatment of 1H-thieno[3,2-d][1,3]oxazine-2,4-dione with different natural alpha-amino acids. |
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