Microwave-assisted in situ deprotection and ω-methoxylation of TMS-protected aryl alkynes |
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Authors: | Jenny WettergrenAlexander B.E. Minidis |
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Affiliation: | Medicinal Chemistry, Local Discovery CNS & Pain Control, AstraZeneca R&D Södertälje, SE-151 85 Södertälje, Sweden |
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Abstract: | Using microwave technology, rapid ω-methoxylation of aryl alkynes is possible. |
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