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In silico ADME/Tox: why models fail
Authors:Stouch Terry R  Kenyon James R  Johnson Stephen R  Chen Xue-Qing  Doweyko Arthur  Li Yi
Institution:(1) Department of Macromolecular Structure, Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton, NJ, USA;(2) Non-clinical Biostatistics, Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton, NJ, USA;(3) Preclinical Optimization, Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton, NJ, USA
Abstract:
Keywords:ADME  QSAR  Validation  Drug Design  Solubility  HERG  Permeation  2D6  In silico
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